{"id":1405025,"date":"2024-08-19T15:31:08","date_gmt":"2024-08-19T13:31:08","guid":{"rendered":"https:\/\/dnaera.com\/hu\/?p=1405025"},"modified":"2024-10-22T12:05:25","modified_gmt":"2024-10-22T10:05:25","slug":"tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny","status":"publish","type":"post","link":"https:\/\/dnaera.com\/hu\/blog\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\/","title":{"rendered":"Tioguan\u00edn \u2013 mal\u00fd bojovn\u00edk, ktor\u00e9ho moc ovplyv\u0148uj\u00fa g\u00e9ny"},"content":{"rendered":"\n<p><em><em>Viete si predstavi\u0165 molekulu tak mal\u00fa, \u017ee ju nevid\u00edte, ale tak siln\u00fa, \u017ee dok\u00e1\u017ee zmeni\u0165 \u017eivot pacienta s\u00a0onkologick\u00fdm ochoren\u00edm? Tioguan\u00edn je presne takou molekulou \u2013 nen\u00e1padn\u00fd a \u00fa\u010dinn\u00fd hrdina v boji proti rakovine. Aby sme v\u0161ak zabezpe\u010dili jeho maxim\u00e1lnu \u00fa\u010dinnos\u0165 a minimalizovali riziko ne\u017eiad\u00facich \u00fa\u010dinkov, je nevyhnutn\u00e9 pochopi\u0165, ako pr\u00edtomnos\u0165 r\u00f4znych genetick\u00fdch variantov v\u00a0na\u0161ej DNA ovplyv\u0148uje jeho metabolizmus.<\/em><\/em><\/p>\n\n\n\n<h2 class=\"wp-block-heading\"><strong><strong><strong><strong><strong><strong><strong><strong>O ak\u00e9 lie\u010divo ide a ako \u00fa\u010dinkuje?<\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/h2>\n\n\n\n<p>Tioguan\u00edn je syntetick\u00e9 lie\u010divo patriace do skupiny tiopur\u00ednov so schopnos\u0165ou p\u00f4sobi\u0165 proti n\u00e1dorom a\u00a0potl\u00e1\u010da\u0165 imunitn\u00fd syst\u00e9m. V\u010faka svojej molekul\u00e1rnej \u0161trukt\u00fare p\u00f4sob\u00ed na \u00farovni DNA t\u00fdm, \u017ee zabra\u0148uje synt\u00e9ze nukleov\u00fdch kysel\u00edn, \u010do vedie k zastaveniu delenia rakovinov\u00fdch buniek. Tento proces efekt\u00edvne nar\u00fa\u0161a ich schopnos\u0165 mno\u017ei\u0165 sa, \u010d\u00edm prispieva k ich postupn\u00e9mu zni\u010deniu.\u00a0<\/p>\n\n\n\n<h2 class=\"wp-block-heading\"><strong><strong><strong><strong><strong><strong><strong><strong>Na \u010do sa pou\u017e\u00edva?<\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/h2>\n\n\n\n<p>V\u010faka svojej schopnosti zacieli\u0165 a eliminova\u0165 r\u00fdchlo sa deliace bunky sa tioguan\u00edn vyu\u017e\u00edva prim\u00e1rne pri lie\u010dbe onkologick\u00fdch ochoren\u00ed, konkr\u00e9tne ak\u00fatnej myeloidnej leuk\u00e9mie.\u00a0<\/p>\n\n\n\n<h2 class=\"wp-block-heading\"><strong><strong><strong><strong><strong><strong><strong><strong>Nie ka\u017ed\u00fd metabolizuje toto lie\u010divo rovnako r\u00fdchlo. Ak\u00fd to m\u00f4\u017ee ma\u0165 dopad?<\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/h2>\n\n\n\n<p>V s\u00favislosti s metabolizmom tioguan\u00ednu, ale aj in\u00fdch lie\u010div, sa be\u017ene pou\u017e\u00edvaj\u00fa pojmy:<\/p>\n\n\n\n<ul class=\"wp-block-list\">\n<li>\u0161tandardn\u00fd metaboliz\u00e9r,\u00a0<\/li>\n<\/ul>\n\n\n\n<ul class=\"wp-block-list\">\n<li>slab\u0161\u00ed metaboliz\u00e9r,<\/li>\n<\/ul>\n\n\n\n<ul class=\"wp-block-list\">\n<li>slab\u00fd metaboliz\u00e9r.<\/li>\n<\/ul>\n\n\n\n<p>Tioguan\u00edn je prolie\u010divo, ktor\u00e9 sa po vstupe do buniek premie\u0148a na akt\u00edvne metabolity schopn\u00e9 p\u00f4sobi\u0165 na rakovinov\u00e9 bunky za\u010dlenen\u00edm do DNA. Hoci s\u00fa tieto akt\u00edvne metabolity \u00fa\u010dinn\u00e9 v&nbsp;boji proti rakovine, m\u00f4\u017eu by\u0165 z\u00e1rove\u0148 toxick\u00e9 pre zdrav\u00e9 bunky a&nbsp;vyvola\u0165 tak ne\u017eiad\u00face \u00fa\u010dinky. G\u00e9ny TPMT a&nbsp;NUDT15 zabezpe\u010duj\u00fa tvorbu enz\u00fdmov d\u00f4le\u017eit\u00fdch pri&nbsp;inaktiv\u00e1cii t\u00fdchto toxick\u00fdch metabolitov v snahe&nbsp;zabezpe\u010di\u0165 rovnov\u00e1hu medzi \u00fa\u010dinnos\u0165ou lie\u010diva a&nbsp;jeho toxicitou. Pr\u00edtomnos\u0165 ur\u010dit\u00fdch genetick\u00fdch variantov v&nbsp;t\u00fdchto g\u00e9noch m\u00e1 za n\u00e1sledok tvorbu enz\u00fdmov so zn\u00ed\u017eenou, popr\u00edpade ch\u00fdbaj\u00facou aktivitou, \u010d\u00edm sa u&nbsp;pacienta zvy\u0161uje riziko rozvoja ne\u017eiad\u00facich \u00fa\u010dinkov a&nbsp;toxicity.<\/p>\n\n\n\n<h2 class=\"wp-block-heading\"><strong><strong><strong><strong><strong><strong><strong><strong><strong>Ak\u00e1 je v\u00fdhoda poznania genetickej predispoz\u00edcie?<\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/h2>\n\n\n\n<p>Poznanie genetickej predispoz\u00edcie pre metabolizmus tioguan\u00ednu je d\u00f4le\u017eitou inform\u00e1ciou pre lek\u00e1ra, \u010di lek\u00e1rnika, s\u00a0ktor\u00fdm v\u00a0pr\u00edpade potreby m\u00f4\u017eete lep\u0161ie a\u00a0r\u00fdchlej\u0161ie optimalizova\u0165 u\u017e\u00edvanie tohto lie\u010diva a\u00a0predch\u00e1dza\u0165 tak vzniku ne\u017eiaducich \u00fa\u010dinkov.<\/p>\n\n\n\n<figure class=\"wp-block-image size-large\"><img fetchpriority=\"high\" decoding=\"async\" width=\"1024\" height=\"358\" src=\"https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog-1024x358.png\" alt=\"\" class=\"wp-image-1405027\" srcset=\"https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog-1024x358.png 1024w, https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog-300x105.png 300w, https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog-768x269.png 768w, https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog-600x210.png 600w, https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog.png 1200w\" sizes=\"(max-width: 1024px) 100vw, 1024px\" \/><\/figure>\n\n\n\n<h2 class=\"wp-block-heading\"><strong><strong><strong><strong><strong><strong><strong><strong>Nov\u00fd v\u00fdsledok anal\u00fdzy<\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/strong><\/h2>\n\n\n\n<p><a href=\"https:\/\/app.dnaera.sk\/sign-in?&amp;lng=sk\" target=\"_blank\" rel=\"noreferrer noopener\">Prihl\u00e1ste sa do svojich v\u00fdsledkov.<\/a> Nov\u00e1 predispoz\u00edcia je odteraz zadarmo dostupn\u00e1 pre v\u0161etk\u00fdch na\u0161ich z\u00e1kazn\u00edkov. Z\u00e1rove\u0148 ju bude ma\u0165 vo svojej anal\u00fdze ka\u017ed\u00fd bud\u00faci z\u00e1kazn\u00edk, ktor\u00fd vst\u00fapi do sveta DNA s <a href=\"https:\/\/dnaera.com\/hu\/produkt\/dna-complex-test\/\" target=\"_blank\" rel=\"noreferrer noopener\">DNA Complex testom<\/a> alebo <a href=\"https:\/\/dnaera.com\/hu\/produkt\/dna-health-test\/\" target=\"_blank\" rel=\"noreferrer noopener\">DNA Health testom<\/a>. Spoznajte svoje predispoz\u00edcie aj vy.<\/p>\n\n\n\n<p><strong>Zdroje<\/strong>:&nbsp;<\/p>\n\n\n\n<ol class=\"wp-block-list\">\n<li class=\"has-small-font-size\">Wang, S., Yuan, X. H., Wang, S. Q., Zhao, W., Chen, X. B., &amp; Yu, B. (2021). FDA-approved pyrimidine-fused bicyclic heterocycles for cancer therapy: Synthesis and clinical application. European Journal of Medicinal Chemistry, 214, 113218.<\/li>\n\n\n\n<li class=\"has-small-font-size\">Goh, L. L., Lim, C. W., Leong, K. P., &amp; Ong, K. H. (2022). TPMT and NUDT15 testing for thiopurine therapy: a major tertiary hospital experience and lessons learned. Frontiers in Pharmacology, 13, 837164.<\/li>\n\n\n\n<li class=\"has-small-font-size\"><a href=\"https:\/\/www.cancer.gov\/types\/leukemia\/patient\/adult-aml-treatment-pdq\">https:\/\/www.cancer.gov\/types\/leukemia\/patient\/adult-aml-treatment-pdq<\/a><\/li>\n<\/ol>\n","protected":false},"excerpt":{"rendered":"<p>Viete si predstavi\u0165 molekulu tak mal\u00fa, \u017ee ju nevid\u00edte, ale tak siln\u00fa, \u017ee dok\u00e1\u017ee zmeni\u0165 \u017eivot pacienta s\u00a0onkologick\u00fdm ochoren\u00edm? Tioguan\u00edn je presne takou molekulou \u2013 nen\u00e1padn\u00fd a \u00fa\u010dinn\u00fd hrdina v boji proti rakovine. Aby sme v\u0161ak zabezpe\u010dili jeho maxim\u00e1lnu \u00fa\u010dinnos\u0165 a minimalizovali riziko ne\u017eiad\u00facich \u00fa\u010dinkov, je nevyhnutn\u00e9 pochopi\u0165, ako pr\u00edtomnos\u0165 r\u00f4znych genetick\u00fdch variantov v\u00a0na\u0161ej DNA [&hellip;]<\/p>\n","protected":false},"author":869,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_acf_changed":false,"content-type":"","inline_featured_image":false,"footnotes":""},"categories":[1],"tags":[58,59,111,63,30],"place-taxonomy":[],"class_list":["post-1405025","post","type-post","status-publish","format-standard","hentry","category-uncategorized-sk","tag-dna-analyza","tag-dna-test","tag-predispozicia","tag-zaujimavosti","tag-zdravie"],"acf":[],"views":2016,"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Tioguan\u00edn \u2013 mal\u00fd bojovn\u00edk, ktor\u00e9ho moc ovplyv\u0148uj\u00fa g\u00e9ny - DNA ERA HU<\/title>\n<meta name=\"description\" content=\"Viete si predstavi\u0165 molekulu tak mal\u00fa, \u017ee ju nevid\u00edte, ale tak siln\u00fa, \u017ee dok\u00e1\u017ee zmeni\u0165 \u017eivot pacienta s\u00a0onkologick\u00fdm ochoren\u00edm? Tioguan\u00edn je presne takou molekulou \u2013 nen\u00e1padn\u00fd a \u00fa\u010dinn\u00fd hrdina v boji proti rakovine.\" \/>\n<meta name=\"robots\" content=\"noindex, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<meta property=\"og:locale\" content=\"hu_HU\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Tioguan\u00edn \u2013 mal\u00fd bojovn\u00edk, ktor\u00e9ho moc ovplyv\u0148uj\u00fa g\u00e9ny\" \/>\n<meta property=\"og:description\" content=\"Viete si predstavi\u0165 molekulu tak mal\u00fa, \u017ee ju nevid\u00edte, ale tak siln\u00fa, \u017ee dok\u00e1\u017ee zmeni\u0165 \u017eivot pacienta s\u00a0onkologick\u00fdm ochoren\u00edm? Tioguan\u00edn je presne takou molekulou \u2013 nen\u00e1padn\u00fd a \u00fa\u010dinn\u00fd hrdina v boji proti rakovine.\" \/>\n<meta property=\"og:url\" content=\"https:\/\/dnaera.com\/hu\/blog\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\/\" \/>\n<meta property=\"og:site_name\" content=\"DNA ERA HU\" \/>\n<meta property=\"article:published_time\" content=\"2024-08-19T13:31:08+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2024-10-22T10:05:25+00:00\" \/>\n<meta name=\"author\" content=\"filipjakubovie\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:image\" content=\"https:\/\/dnaera.com\/hu\/wp-content\/uploads\/sites\/7\/2024\/08\/SK-tiog.png\" \/>\n<meta name=\"twitter:label1\" content=\"Szerz\u0151:\" \/>\n\t<meta name=\"twitter:data1\" content=\"filipjakubovie\" \/>\n\t<meta name=\"twitter:label2\" content=\"Becs\u00fclt olvas\u00e1si id\u0151\" \/>\n\t<meta name=\"twitter:data2\" content=\"3 perc\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\\\/\\\/schema.org\",\"@graph\":[{\"@type\":\"Article\",\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/#article\",\"isPartOf\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/\"},\"author\":{\"name\":\"filipjakubovie\",\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/#\\\/schema\\\/person\\\/2ccfc4fabdb15105d6234432c5cfa85e\"},\"headline\":\"Tioguan\u00edn \u2013 mal\u00fd bojovn\u00edk, ktor\u00e9ho moc ovplyv\u0148uj\u00fa g\u00e9ny\",\"datePublished\":\"2024-08-19T13:31:08+00:00\",\"dateModified\":\"2024-10-22T10:05:25+00:00\",\"mainEntityOfPage\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/\"},\"wordCount\":588,\"publisher\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/#organization\"},\"image\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/#primaryimage\"},\"thumbnailUrl\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/wp-content\\\/uploads\\\/sites\\\/7\\\/2024\\\/08\\\/SK-tiog-1024x358.png\",\"keywords\":[\"DNA anal\u00fdza\",\"DNA test\",\"predispozicia\",\"zauj\u00edmavosti\",\"zdravie\"],\"articleSection\":[\"Uncategorized @sk\"],\"inLanguage\":\"hu\"},{\"@type\":\"WebPage\",\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/\",\"url\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/\",\"name\":\"Tioguan\u00edn \u2013 mal\u00fd bojovn\u00edk, ktor\u00e9ho moc ovplyv\u0148uj\u00fa g\u00e9ny - DNA ERA HU\",\"isPartOf\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/#website\"},\"primaryImageOfPage\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/#primaryimage\"},\"image\":{\"@id\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/blog\\\/tioguanin-maly-bojovnik-ktoreho-moc-ovplyvnuju-geny\\\/#primaryimage\"},\"thumbnailUrl\":\"https:\\\/\\\/dnaera.com\\\/hu\\\/wp-content\\\/uploads\\\/sites\\\/7\\\/2024\\\/08\\\/SK-tiog-1024x358.png\",\"datePublished\":\"2024-08-19T13:31:08+00:00\",\"dateModified\":\"2024-10-22T10:05:25+00:00\",\"description\":\"Viete si predstavi\u0165 molekulu tak mal\u00fa, \u017ee ju nevid\u00edte, ale tak siln\u00fa, \u017ee dok\u00e1\u017ee zmeni\u0165 \u017eivot pacienta s\u00a0onkologick\u00fdm ochoren\u00edm? 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